O le fualaau faasaina "Buserelin Long" o se analogue gaosi o le hormone faalenatura GnRH. O le faagaoioiga o lenei meafaigaluega e saʻo faatauva noatia e receptors sela ma faateleina tumau mulimuli ane pituitary i tulaga o feusuaiga steroids i plasma, lea na iu lava ina taunuu i le atoatoa blockage o le mea ua taʻua o gonadotropic galuega tauave pituitary. O se taunuuga o le fualaau faasaina "Buserelin Long" ua tuuina saʻo taofia tuufaatasia hormone i le gonads, lea e faaalia ia lava e avea o se faaitiitia o tulaga testosterone (indices e faapipii-castration) i alii ma faaitiitia toto estradiol e faapipii-menopausal uiga i gasegase fafine. I le tulaga muamua e mafai ona tatou talanoa e uiga i castration pharmacological, i le lona lua - i postmenopausal po ovariectomy.
ua faamatuu le vailaau i se taimi o se lyophilizate faapitoa fuafuaina e saunia se slurry. Le tuufaatasiga o lenei sauniuniga o se elemene autu e aofia ai e uiga i 4 mg acetate buserelin. vaega o ausilali e aofia sodium carmellose, o se copolymer o glycolic ma dl-lactic acid, polysorbate-80 ma d-mannitol.
E tusa ai ma le faaaogaina o le fualaau faasaina, o le sui e tofia "Buserelin Long" mo le togafitiga o le fatafata kanesa ma hormone-faalagolago kanesa prostate. I le faaopoopo atu, e mafai ona faaaogaina ai lenei fualaau faasaina i le taimi o le togafitiga o endometriosis. Mo le togafitia o fibroids ma le mauaina o fanau uterine (e ala i le polokalama IVF) E tatau foi ona e amata faaaogaina le fualaau faasaina "Buserelin-Long". Iloiloga o fomai molimau atu e uiga i le taunuuga lelei o lona faaaogaina mo le togafitia o faiga hyperplastic endometrial.
Afai tatou te talanoa e uiga i le contraindications autu i le faaaogāina, ona faaaoga lea o lenei vailaau contraindicated tonu mo tagata ma acetate buserelin le le faapalepale o tagata taitoatasi, faapea foi ma so o se isi o ona vaega e lagolago ai. I le faaopoopo atu, contraindications aofia maitaga ma lactation.
Eseese, e tatau ona fai e uiga i le aafiaga itu talafeagai o le faaaogaina o tupe "Buserelin-Long", e pei ona mafai ona avea, mo se faataitaiga, o le mafuaaga o urticaria, angioneurotic edema ma hyperemia. I le gata i lea, atonu ei ai tulaga e pei o demineralization, faasoesa moe, ulu tiga ma le faanoanoa. I oo gasegase fafine tiga lona manava, suiga i libido, faateleina afuafu tetele, menstrualnopodobnye tafetotoi ma faʻamago o le mucosa vaginal ona o le faaaogaina o fualaau faasaina e gaosia "Buserelin-Long". ua mafua fesootai Itu aafiaga i tagata ma le exacerbation o faamaʻi faavae, faatumauina urinary, gynecomastia, ma le "fula fatugao." I le faaopoopo atu, e mafai ona faailogaina faaitiitia o potency, faateleina afuafu tetele, maso vaivaiga i le tiga pito ma ivi. O se vaega toaitiiti o gasegase e mafai ona oo i ai tali e pei o le faaletonu diarrheal , ma embolism chronic.